SCHEMBL7943655

SCHEMBL7943655

CCOC(=O)c1cn2c(n1)CN=C(c1ccccn1)c1cc(Br)ccc1-2

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 11/20 0.55
GABRA3 P34903 9/20 0.55
GABRA2 P47869 9/20 0.55
GABRA1 P14867 6/20 0.55
GABRB2 P47870 5/20 0.55
GABRG2 P18507 11/20 0.53
GABRB3 P28472 11/20 0.53
ADRA1A P35348 1/20 0.43
GABRA6 Q16445 3/20 0.41
CYP1A2 P05177 1/20 0.40
GABRA4 P48169 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369039 0.86 GABRA5 (0.53) GABRA5GABRA3GABRA2GABRA1GABRB2
SCHEMBL3415178 0.81 GABRG2 (0.77) GABRA5GABRA3GABRA2GABRA1GABRB2
SCHEMBL7380104 0.80 GABRA3 (0.58) GABRA5GABRA3GABRA2GABRA1GABRB2
SCHEMBL7312677 0.79 GABRA5 (0.57) GABRA5GABRA3GABRA2GABRA1GABRB2
SCHEMBL11731330 0.74 GABRA3 (0.64) GABRA5GABRA3GABRA2GABRA1GABRB2
SCHEMBL7431448 0.73 GABRA3 (0.66) GABRA5GABRA3GABRA2GABRA1GABRB2
SCHEMBL11709742 0.72 GABRA3 (0.66) GABRA5GABRA3GABRA2GABRA1GABRB2
SCHEMBL19368522 0.72 GABRG2 (0.58) GABRA5GABRA3GABRA2GABRA1GABRG2
SCHEMBL3142139 0.72 GABRG2 (0.58) GABRA5GABRA3GABRA2GABRA1GABRG2
SCHEMBL7722605 0.72 GABRG2 (0.58) GABRA5GABRA3GABRA2GABRA1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174881-B1 USED AS ANXIOLYTIC AND/OR ANTICONVULSANT AND/OR MUSCLE RELAXANT AGENTS; SEDATIVES OR HYPNOSIS; WATER-SOLUBLE AMINE SALTS; FAST-ACTING HOFFMAN-LA ROCHE INC. 2001-01-16 US disclosed