SCHEMBL7944647

SCHEMBL7944647

Cc1cccc(-c2nc3c(N)ccnc3n(C(C)C)c2=O)c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTOR P42345 7/20 0.53
SRC P12931 3/20 0.44
XDH P47989 2/20 0.38
PDE4B Q07343 1/20 0.38
ABL1 P00519 1/20 0.38
NR1I2 O75469 1/20 0.37
EGFR P00533 1/20 0.37
ADRA2A P08913 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
TBXA2R P21731 1/20 0.37
PTGS2 P35354 1/20 0.37
OPRD1 P41143 1/20 0.37
PDE4D Q08499 1/20 0.37
TLR8 Q9NR97 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPK14 Q16539 1/20 0.36
PIK3CD O00329 1/20 0.36
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7946228 0.88 MTOR (0.48) MTOR
SCHEMBL7947069 0.85 MTOR (0.48) MTORSRCXDHABL1EGFR
SCHEMBL7947571 0.82 PDE4B (0.47) MTORSRCPDE4BABL1ADORA3
SCHEMBL7947917 0.80 PDE4B (0.51) MTORSRCPDE4BABL1ADORA3
SCHEMBL7938164 0.78 PDE4B (0.42) MTORSRCPDE4BABL1MAPK14
SCHEMBL7946067 0.78 PDE4B (0.57) PDE4BPDE4DTLR8KMT2AMAPK14
SCHEMBL7945984 0.78 CYP1A2 (0.51) PDE4BKMT2A
SCHEMBL7947972 0.72 CYP1A2 (0.57) PDE4BKMT2A
SCHEMBL7944713 0.70 CYP1A2 (0.47) PDE4BKMT2A
SCHEMBL7938047 0.70 CYP1A2 (0.56) MTORSRCABL1EGFRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed