SCHEMBL7945652

SCHEMBL7945652

COC(=O)c1cc2c3c(cc(O)c2[nH]1)N(C(=O)c1cc2cc(OC)ccc2[nH]1)CC3CCl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HRH4 Q9H3N8 1/20 0.42
AKR1C3 P42330 1/20 0.41
XDH P47989 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
PDGFRB P09619 2/20 0.40
PDGFRA P16234 1/20 0.40
DRD2 P14416 2/20 0.40
DRD3 P35462 2/20 0.40
FLT3 P36888 4/20 0.39
ADH1A P07327 1/20 0.39
KIT P10721 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7959056 0.94 KMT2A (0.45) NPC1RAB9AHRH4MEN1KMT2A
SCHEMBL7945647 0.89 ADH1A (0.45) KDM4ENPC1RAB9ALMNAL3MBTL1
SCHEMBL20991116 0.88 HRH4 (0.47) KDM4ENPC1RAB9AALDH1A1HRH4
SCHEMBL6517364 0.86 ADH1A (0.53) KDM4ENPC1RAB9AHRH4AKR1C3
SCHEMBL6517359 0.86 ADH1A (0.53) KDM4ENPC1RAB9AHRH4AKR1C3
SCHEMBL14669320 0.85 NPC1 (0.41) KDM4ENPC1RAB9ALMNAAKR1C3
SCHEMBL6620418 0.85 NPC1 (0.41) KDM4ENPC1RAB9ALMNAAKR1C3
SCHEMBL7952123 0.85 HRH4 (0.44) NPC1RAB9AHRH4MEN1KMT2A
SCHEMBL5864982 0.83 DRD2 (0.44) KDM4EHRH4AKR1C3MEN1KMT2A
SCHEMBL30360049 0.83 P4HB (0.51) KDM4ERAB9AALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281354-B1 ANTIBIOTICS; ANTITUMOR AGENTS THE SCRIPPS RESEARCH INSTITUTE 2001-08-28 US disclosed