SCHEMBL7945866

SCHEMBL7945866

[CH2]c1ccc(OCCCN2CCN(C)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.66
NPC1 O15118 1/20 0.66
ALDH1A1 P00352 2/20 0.65
USP2 O75604 2/20 0.65
HPGD P15428 1/20 0.65
HRH3 Q9Y5N1 6/20 0.62
DRD3 P35462 1/20 0.61
MAPK1 P28482 3/20 0.54
CYP1A2 P05177 1/20 0.54
CHRM2 P08172 1/20 0.54
CHRM1 P11229 1/20 0.54
HTR2A P28223 1/20 0.54
SCN1A P35498 1/20 0.54
HTR2B P41595 1/20 0.54
KCNH2 Q12809 1/20 0.54
SCN2A Q99250 1/20 0.54
SIGMAR1 Q99720 1/20 0.54
SCN3A Q9NY46 1/20 0.54
LTA4H P09960 1/20 0.54
MEN1 O00255 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7954349 0.92 LTA4H (0.63) RAB9ANPC1ALDH1A1USP2HPGD
SCHEMBL23291197 0.87 HRH3 (0.68) RAB9ANPC1ALDH1A1USP2HPGD
SCHEMBL7956510 0.86 HRH3 (0.72) HRH3KCNH2MEN1KMT2A
SCHEMBL2827360 0.85 HRH3 (0.75) HRH3KCNH2
SCHEMBL8360712 0.85 RAB9A (0.68) RAB9ANPC1ALDH1A1USP2HPGD
SCHEMBL10817906 0.83 RAB9A (0.76) RAB9ANPC1ALDH1A1USP2HPGD
SCHEMBL12359053 0.83 USP2 (0.91) RAB9ANPC1ALDH1A1USP2HPGD
SCHEMBL16301445 0.83 RAB9A (0.66) RAB9ANPC1ALDH1A1USP2HPGD
SCHEMBL76269 0.83 RAB9A (0.66) RAB9ANPC1ALDH1A1USP2HPGD
SCHEMBL19091219 0.83 RAB9A (0.79) RAB9ANPC1ALDH1A1USP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6297274-B1 SUBSTITUTED 5-HYDROXYFURANONES WARNER-LAMBERT COMPANY 2001-10-02 US claimed
WO-1997037985-A1 NONPEPTIDE ENDOTHELIN ANTAGONISTS WITH INCREASED WATER SOLUBILITY WARNER-LAMBERT COMPANY (US) 1997-10-16 WO claimed
US-6297274-B1 SUBSTITUTED 5-HYDROXYFURANONES WARNER-LAMBERT COMPANY 2001-10-02 US disclosed
WO-1997037985-A1 NONPEPTIDE ENDOTHELIN ANTAGONISTS WITH INCREASED WATER SOLUBILITY WARNER-LAMBERT COMPANY (US) 1997-10-16 WO disclosed