SCHEMBL7946084

SCHEMBL7946084

CCCn1c(=O)c(C)nc2c(N)cc(NCCO)nc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.37
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 2/20 0.36
IKBKB O14920 1/20 0.35
ALDH1A1 P00352 5/20 0.34
CYP1A2 P05177 2/20 0.34
HSD17B10 Q99714 2/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
PDE4A P27815 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
CDK1 P06493 1/20 0.34
ADORA2B P29275 3/20 0.33
TLR9 Q9NR96 1/20 0.33
ADORA1 P30542 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7937861 0.85 TLR9 (0.35) HRH4CYP2D6CYP2C19IKBKBPDE4A
SCHEMBL7943760 0.79 CD38 (0.37) CYP2C19ALDH1A1CYP1A2HSD17B10KDM4E
SCHEMBL7945503 0.76 TLR9 (0.37) CYP2D6CYP2C19ALDH1A1CYP1A2HSD17B10
SCHEMBL7937747 0.72 HSF1 (0.35) CYP2D6ALDH1A1CYP1A2HSD17B10CYP2C9
SCHEMBL7943995 0.68 HSF1 (0.36) CYP2D6CYP2C19ALDH1A1CYP1A2HSD17B10
SCHEMBL7944093 0.66 STIM1 (0.38) ALDH1A1KDM4EADORA2BTLR9ADORA1
SCHEMBL6118631 0.60 CYP2D6 (0.51) HRH4CYP2D6CYP2C19IKBKBALDH1A1
SCHEMBL8130946 0.60 PDE4A (0.56) HSD17B10HPGDPDE4APDE4BPDE4C
SCHEMBL20470731 0.59 CYP2D6 (0.46) HRH4CYP2D6CYP2C19IKBKBALDH1A1
SCHEMBL8132409 0.57 PDE4A (0.50) IKBKBCYP1A2HSD17B10PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed