SCHEMBL7943760

SCHEMBL7943760

CCCn1c(=O)c(C)nc2c(N)cc(NCc3c(F)cccc3F)nc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD38 P28907 1/20 0.37
ADORA2B P29275 3/20 0.36
ALDH1A1 P00352 3/20 0.36
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
POLB P06746 1/20 0.35
USP2 O75604 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
KDM4E B2RXH2 3/20 0.33
TP53 P04637 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
RAB9A P51151 1/20 0.33
STIM1 Q13586 1/20 0.33
ORAI1 Q96D31 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7944093 0.87 STIM1 (0.38) CD38ADORA2BALDH1A1CCNT1CDK9
SCHEMBL7937752 0.82 ADORA2A (0.39) ADORA2BALDH1A1CCNT1CDK9POLB
SCHEMBL7946084 0.79 HRH4 (0.37) ADORA2BALDH1A1POLBCYP1A2CYP2C19
SCHEMBL3227728 0.70 SCN8A (0.37) CD38ALDH1A1CCNT1CDK9CYP1A2
SCHEMBL7945503 0.70 TLR9 (0.37) ADORA2BALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL7937861 0.67 TLR9 (0.35) ADORA2BCYP2C19TMIGD3ADORA2AADORA1
SCHEMBL7943995 0.64 HSF1 (0.36) ALDH1A1USP2CYP1A2CYP3A4CYP2C19
SCHEMBL7937747 0.63 HSF1 (0.35) ALDH1A1USP2CYP1A2CYP3A4HSD17B10
SCHEMBL7938416 0.60 CYP1A2 (0.50) ALDH1A1USP2CYP1A2CYP3A4CYP2C19
SCHEMBL7947917 0.58 PDE4B (0.51) ADORA2BALDH1A1USP2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed