SCHEMBL7944912

SCHEMBL7944912

CCCOc1cc(-c2ccc(C#N)cc2)ccc1CBr

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HRH3 Q9Y5N1 7/20 0.39
MMP2 P08253 5/20 0.38
ALDH1A1 P00352 3/20 0.37
HPGD P15428 3/20 0.37
HRH2 P25021 3/20 0.36
HRH1 P35367 3/20 0.36
MMP3 P08254 3/20 0.36
KDM4E B2RXH2 3/20 0.36
ICMT O60725 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MMP1 P03956 1/20 0.35
MMP9 P14780 1/20 0.35
MMP13 P45452 1/20 0.35
PTGER4 P35408 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7943319 0.86 MMP2 (0.40) TSHRHSD17B10HRH3MMP2ALDH1A1
SCHEMBL7946267 0.78 PPARD (0.41)
SCHEMBL7943031 0.77 ERN1 (0.49) TSHRHSD17B10HRH3MMP2ALDH1A1
SCHEMBL27001729 0.77 CYP19A1 (0.41) MMP2ALDH1A1ICMT
SCHEMBL5405545 0.76 TRPV4 (0.54) HSD17B10ALDH1A1HPGD
SCHEMBL12736275 0.75 MMP2 (0.60) HRH3MMP2ALDH1A1HPGDHRH2
SCHEMBL2462665 0.75 MMP2 (0.60) HRH3MMP2ALDH1A1HPGDHRH2
SCHEMBL6098475 0.75 ERN1 (0.50) TSHRHSD17B10HRH3MMP2ALDH1A1
SCHEMBL7984620 0.74 CYP19A1 (0.54) TSHRHSD17B10HPGDMMP13
SCHEMBL7361936 0.74 CSNK2A1 (0.42) ALDH1A1HPGDKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015653-A1 PYRIMIDINE DERIVATIVES AS ACTIVATORS OF SOLUBLE GUANYLATE CYCLASE SMITHKLINE BEECHAM CORPORATION (US) 2010-02-11 WO disclosed
WO-2009071504-A1 2,6-DISUBSTITUTED PYRIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-11 WO disclosed