SCHEMBL7946362

SCHEMBL7946362

NC(=O)c1cc(-c2ccncc2)n2c1CCCC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 10/20 0.50
CDK9 P50750 1/20 0.50
CHUK O15111 2/20 0.41
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
CASP1 P29466 1/20 0.39
GAA P10253 1/20 0.38
TBK1 Q9UHD2 1/20 0.38
CYP11B2 P19099 2/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
IKBKB O14920 1/20 0.36
IKBKE Q14164 1/20 0.36
PKMYT1 Q99640 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2157288 0.85 MKNK1 (0.46) CYP2C9GAACYP11B2
SCHEMBL7953665 0.81 MKNK1 (0.47) KMT2ACYP11B2
SCHEMBL2158167 0.80 SIRT3 (0.46) CDC7CDK9MEN1CYP1A2CYP3A4
SCHEMBL7955655 0.75 WNT1 (0.35) CDC7CDK9MEN1KMT2AGAA
SCHEMBL7960316 0.75 KDM4A (0.35) CDC7CDK9MEN1KMT2AGAA
SCHEMBL7946519 0.75 PLAU (0.41) CYP3A4GAA
SCHEMBL7957597 0.75 HPGD (0.37) GAAIKBKB
SCHEMBL7954859 0.75 MKNK1 (0.43) GAA
SCHEMBL7953705 0.73 CYP2C9 (0.43) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7953580 0.72 CYP11B1 (0.37) MEN1CYP2C19KMT2ACYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194426-B1 CONTROLLING TUMOR NECROSIS FACTOR RHONA-POULENC RORER S.A. (FR) 2001-02-27 US disclosed
EP-0833635-A1 NOVEL USE FOR PYRROLE DERIVATIVES Aventis Pharma S.A. (FR) 1998-04-08 EP disclosed
WO-1997000073-A1 NOVEL USE FOR PYRROLE DERIVATIVES RHONE-POULENC RORER S.A. (FR) 1997-01-03 WO disclosed