SCHEMBL7947307

SCHEMBL7947307

N#Cc1ccccc1S(=O)(=O)Nc1ccc(N2CCN(c3ccncc3)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 4/20 0.51
ALDH1A1 P00352 4/20 0.50
MAPT P10636 4/20 0.50
KMT2A Q03164 3/20 0.50
GFER P55789 2/20 0.50
GAA P10253 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HSPD1 P10809 1/20 0.47
PTPN2 P17706 1/20 0.47
PTPN1 P18031 1/20 0.47
PTPN5 P54829 1/20 0.47
HSPE1 P61604 1/20 0.47
BRD1 O95696 1/20 0.47
BRPF1 P55201 1/20 0.47
SLC40A1 Q9NP59 1/20 0.46
LMNA P02545 2/20 0.45
KDM4E B2RXH2 1/20 0.45
SGK1 O00141 1/20 0.44
PKLR P30613 1/20 0.44
HTR6 P50406 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7956237 0.83 GAA (0.44) ALDH1A1KMT2AGAALMNAKDM4E
SCHEMBL96355 0.74 SLC22A12 (0.63) SLC22A12KMT2AHSPD1PTPN2PTPN1
SCHEMBL10682806 0.72 CHKA (0.47) MAPTLMNAHPGD
SCHEMBL10680323 0.72 JAK2 (0.50) ALDH1A1MAPTLMNA
SCHEMBL7954743 0.71 NAMPT (0.59) ALDH1A1MAPTLMNAKDM4EPKLR
SCHEMBL2955815 0.69 PKM (0.63) ALDH1A1KMT2AGAATDP1KDM4E
SCHEMBL6363732 0.68 GFER (0.98) ALDH1A1MAPTKMT2AGFERGAA
SCHEMBL7947310 0.67 MCOLN3 (0.50) SLC22A12GAATDP1KDM4E
SCHEMBL6362807 0.67 GFER (1.00) ALDH1A1MAPTKMT2AGFERGAA
SCHEMBL7956560 0.67 KDM4E (0.65) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313127-B1 FOR THERAPY OF HYPERCHOLESTEROLEMIA OR ATHEROSCLEROSIS ZENECA LIMITED (GB) 2001-11-06 US disclosed
EP-0880501-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997028128-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1997-08-07 WO disclosed