SCHEMBL7947433

SCHEMBL7947433

COc1cc(NC(=S)NC(C)c2ccc(C#N)cc2)c(OC)cc1NC(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.52
MEN1 O00255 4/20 0.52
ALDH1A1 P00352 4/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
MAPT P10636 3/20 0.49
MAPK1 P28482 2/20 0.49
AHR P35869 1/20 0.49
KDM4E B2RXH2 3/20 0.47
GAA P10253 2/20 0.47
EPHX1 P07099 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSD17B10 Q99714 1/20 0.45
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6815737 0.87 ALDH1A1 (0.51) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL7947438 0.83 KMT2A (0.47) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL6811835 0.77 ALDH1A1 (0.53) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL6814533 0.75 ALDH1A1 (0.55) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL19465247 0.73 MEN1 (0.70) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8714750 0.72 MLYCD (0.63) KMT2AMEN1ALDH1A1MAPTAHR
SCHEMBL6812274 0.72 KMT2A (0.54) KMT2AMEN1ALDH1A1CYP2C9CYP2C19
SCHEMBL6814884 0.71 ALDH1A1 (0.51) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL6815741 0.71 KMT2A (0.46) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL31616406 0.70 LMNA (0.61) KMT2AMEN1ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6262082-B1 Diaminopyridine-containing thiourea inhibitors of herpes viruses WYETH 2001-07-17 US disclosed