SCHEMBL7947438

SCHEMBL7947438

COc1cc(N(S)C(=O)NC(C)c2ccc(C#N)cc2)c(OC)cc1NC(=O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.47
MEN1 O00255 5/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPK1 P28482 2/20 0.44
MAPT P10636 2/20 0.44
AHR P35869 1/20 0.44
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 1/20 0.41
POLB P06746 2/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PHGDH O43175 1/20 0.40
GPR139 Q6DWJ6 1/20 0.39
THRB P10828 1/20 0.39
RECQL P46063 1/20 0.39
BLM P54132 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7947433 0.83 KMT2A (0.52) KMT2AMEN1SMN1; SMN2ALDH1A1MAPK1
SCHEMBL6819526 0.78 KMT2A (0.50) KMT2AMEN1SMN1; SMN2ALDH1A1MAPT
SCHEMBL6811843 0.73 ALDH1A1 (0.48) KMT2AMEN1SMN1; SMN2ALDH1A1MAPK1
SCHEMBL6815737 0.71 ALDH1A1 (0.51) KMT2AMEN1SMN1; SMN2ALDH1A1MAPT
SCHEMBL7784293 0.70 KMT2A (0.46) KMT2AMEN1SMN1; SMN2ALDH1A1MAPT
SCHEMBL6815704 0.68 KMT2A (0.50) KMT2AMEN1ALDH1A1
SCHEMBL8714750 0.68 MLYCD (0.63) KMT2AMEN1ALDH1A1MAPTAHR
SCHEMBL6814706 0.67 LMNA (0.41) SMN1; SMN2ALDH1A1MAPTPHGDHL3MBTL1
SCHEMBL6816428 0.67 LMNA (0.41) KMT2ASMN1; SMN2ALDH1A1MAPK1MAPT
SCHEMBL19465247 0.67 MEN1 (0.70) KMT2AMEN1SMN1; SMN2ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6262082-B1 Diaminopyridine-containing thiourea inhibitors of herpes viruses WYETH 2001-07-17 US disclosed