SCHEMBL7947607

SCHEMBL7947607

CC(C)(C)[Si](C)(C)OC1CCN(c2ccncc2Br)C1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 1/20 0.38
CYP46A1 Q9Y6A2 3/20 0.33
IKBKB O14920 2/20 0.33
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32
GBA1 P04062 1/20 0.31
LIPG Q9Y5X9 1/20 0.30
CYP11B2 P19099 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7956455 0.85 ROCK2 (0.37) CA12CA1CA2CA9LIPG
SCHEMBL7958631 0.79 HRH3 (0.43) CYP11B2HRH3
SCHEMBL11907738 0.79 MAPT (0.40)
SCHEMBL4555535 0.79 MAPT (0.40)
SCHEMBL4435998 0.79 MAPT (0.40)
SCHEMBL30784155 0.77 PBRM1 (0.33) GBA1
SCHEMBL30784128 0.77 PBRM1 (0.33) GBA1
SCHEMBL25232014 0.76 CA1 (0.39) CA12CA1CA2CA9LIPG
SCHEMBL30466332 0.76 CA1 (0.39) CA12CA1CA2CA9LIPG
SCHEMBL25277048 0.76 CA1 (0.39) CA12CA1CA2CA9LIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313127-B1 FOR THERAPY OF HYPERCHOLESTEROLEMIA OR ATHEROSCLEROSIS ZENECA LIMITED (GB) 2001-11-06 US disclosed
EP-0880501-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997028128-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1997-08-07 WO disclosed