SCHEMBL7956455

SCHEMBL7956455

CC(C)(C)[Si](C)(C)OC1CCN(c2ccncc2F)C1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 9/20 0.37
PRKG1 Q13976 9/20 0.37
CYP1A2 P05177 2/20 0.36
LIMK2 P53671 1/20 0.36
EHMT2 Q96KQ7 1/20 0.36
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
ACACB O00763 2/20 0.33
LIPG Q9Y5X9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7947607 0.85 RPS6KB1 (0.38) CA12CA1CA2CA9LIPG
SCHEMBL317170 0.82 ROCK2 (0.42) ROCK2PRKG1CYP1A2LIMK2EHMT2
SCHEMBL6544895 0.80 ALDH1A1 (0.41) ACACBLIPG
SCHEMBL7805636 0.80 ALDH1A1 (0.41) ACACBLIPG
SCHEMBL7958631 0.79 HRH3 (0.43) ACACB
SCHEMBL4555535 0.79 MAPT (0.40)
SCHEMBL11907738 0.79 MAPT (0.40)
SCHEMBL4435998 0.79 MAPT (0.40)
SCHEMBL7078416 0.75 ALDH1A1 (0.48)
SCHEMBL7814936 0.75 ALDH1A1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313127-B1 FOR THERAPY OF HYPERCHOLESTEROLEMIA OR ATHEROSCLEROSIS ZENECA LIMITED (GB) 2001-11-06 US disclosed
EP-0880501-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997028128-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1997-08-07 WO disclosed