SCHEMBL7947642

SCHEMBL7947642

Nc1nc(Cc2ccccc2)c2nc(NCCO)nc(Cc3ccccc3)c2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.47
RECQL P46063 1/20 0.46
MCL1 Q07820 1/20 0.46
CDK1 P06493 4/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
CDK2 P24941 2/20 0.43
CDK5 Q00535 2/20 0.43
CCNB2 O95067 1/20 0.43
CCNE2 O96020 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CCNB1 P14635 1/20 0.43
ALOX15 P16050 1/20 0.43
NFKB1 P19838 1/20 0.43
CCNA2 P20248 1/20 0.43
CCNE1 P24864 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4932531 0.79 LTB4R (0.51) RECQLMCL1CDK1KDM4EALDH1A1
SCHEMBL27776002 0.75 LTB4R (0.44) MPOCDK1KDM4EALDH1A1GAA
SCHEMBL11307118 0.72 SLC29A1 (0.45) MPOHTR2BGPR68ADORA2AKMT2A
SCHEMBL168411 0.71 MPO (0.54) MPOCYP1A2CYP3A4CYP2D6SMN1; SMN2
SCHEMBL27393423 0.70 RECQL (0.84) RECQLMCL1CDK5MAPTCDK5R1
SCHEMBL8410920 0.70 NPSR1 (0.68) RECQLMCL1KDM4EALDH1A1GAA
SCHEMBL28198401 0.69 CDK1 (0.51) CDK1KDM4EALDH1A1GAACDK2
SCHEMBL27686623 0.69 CDK1 (0.47) CDK1KDM4EALDH1A1GAACDK2
SCHEMBL7960340 0.69 ALDH1A1 (0.38) RECQLMCL1CDK1KDM4EALDH1A1
SCHEMBL1033545 0.68 KMT2A (0.50) RECQLMCL1CDK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001517226-A 2001-10-02 JP claimed
EP-0971925-A1 PYRIMIDOPYRIMIDINE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 2000-01-19 EP claimed
WO-1998043974-A1 PYRIMIDOPYRIMIDINE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 1998-10-08 WO claimed