SCHEMBL7950574

SCHEMBL7950574

CC(=O)C(OS(=O)(=O)c1ccc(C)cc1)C(N)Cc1cccc(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A1 P43005 2/20 0.42
PLAU P00749 2/20 0.39
PLAT P00750 1/20 0.39
ALDH1A1 P00352 4/20 0.38
HPGD P15428 1/20 0.38
LMNA P02545 1/20 0.36
ROCK2 O75116 1/20 0.36
KMT2A Q03164 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
MAOB P27338 2/20 0.36
PKM P14618 1/20 0.36
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
ADAMTS4 O75173 1/20 0.35
MMP13 P45452 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7950570 0.79 SLC1A1 (0.43) SLC1A1PLAUPLATALDH1A1HPGD
SCHEMBL8770455 0.72 P2RX7 (0.43) ALDH1A1HPGDLMNAKMT2ABCHE
SCHEMBL7961908 0.72 SLC1A1 (0.55) SLC1A1ROCK2KMT2AMAOBPPARG
SCHEMBL7950818 0.72 TDP1 (0.42) ALDH1A1LMNABCHEACHE
SCHEMBL10069421 0.71 SLC1A1 (0.60) SLC1A1ROCK2MAOBPKMPPARG
SCHEMBL21417397 0.71 SLC1A1 (0.60) SLC1A1ROCK2MAOBPKMPPARG
SCHEMBL776918 0.71 ALDH1A1 (0.50) ALDH1A1BCHEACHEMAOBPKM
SCHEMBL10811604 0.70 MMP9 (0.40) ALDH1A1HPGDLMNAKMT2APKM
SCHEMBL5843078 0.69 CYP19A1 (0.46) ALDH1A1LMNAKMT2ABCHEACHE
SCHEMBL7723991 0.69 ALDH1A1 (0.46) ALDH1A1BCHEACHEPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271238-B1 USEFUL IN TREATING AND PREVENTING DISEASES INVOLVING CHYMOTRYPSIN TYPE PROTEASES WHICH ARE RELATED TO ASTHMA, ALLERGY, INFLAMMATIONS, RHEUMATISM, HYPERTENSION, HEART FAILURE, MYOCARDIAL INFARCTION, AND CARDIAC HYPERTROPHY NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-08-07 US disclosed
EP-0936216-A1 NOVEL ACETAMIDE DERIVATIVES AND PROTEASE INHIBITORS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1999-08-18 EP disclosed