SCHEMBL7951653

SCHEMBL7951653

COc1c(C)c[n+]([O-])cc1C

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.33
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12936090 0.73 KDM4E (0.33) ALDH1A1KDM4E
SCHEMBL6841716 0.72 SMN1; SMN2 (0.34) ALDH1A1SMN1; SMN2
SCHEMBL4546154 0.72 HSP90AA1 (0.36) ALDH1A1
SCHEMBL312454 0.70
SCHEMBL8830029 0.69 HSP90AA1 (0.34)
SCHEMBL192045 0.69 HSP90AA1 (0.34)
SCHEMBL5894620 0.69 KDM4E (0.34) ALDH1A1KDM4EMAPK1SMN1; SMN2
SCHEMBL3562505 0.67 GPR84 (0.36) ACHEALDH1A1MAPK1
SCHEMBL20822276 0.67 SOS1 (0.31)
SCHEMBL1044124 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107235961-A A kind of preparation method of esomeprazole 武汉励合生物医药科技有限公司 2017-10-10 CN claimed
CN-107235961-A A kind of preparation method of esomeprazole 武汉励合生物医药科技有限公司 2017-10-10 CN disclosed
CN-103880741-A Preparation method of 2-chloromethyl-3,5-dimethyl-4-alkoxypyridyl-N-oxide ANHUI COSTAR BIO CHEMICAL CO LTD 2014-06-25 CN disclosed
US-6303787-B1 STARTING FROM 4-NITRO-2,3,5-TRIMETHYLPYRIDINE-N-OXIDE AND5-METHOXY-2-MERCAPTO BENZIMIDAZOLE NATCO PHARMA LIMITED (IN) 2001-10-16 US disclosed
EP-1005457-A1 PREPARATION OF PYRIDINE DERIVATIVES Seal Sands Chemicals Limited (GB) 2000-06-07 EP disclosed
WO-1999010326-A1 PREPARATION OF PYRIDINE DERIVATIVES SEAL SANDS CHEMICALS LIMITED (GB) 1999-03-04 WO disclosed
US-5066810-A 3,5-DIMETHYL-4-METHOXYPYRIDINE DERIVATIVES CL PHARMA AKTIENGESELLSCHAFT (AT) 1991-11-19 US disclosed
CN-1042705-A 3,5-dimethyl-4-methoxypyridine derivatization method and be used for the novel intermediate product of this method for making CL PHARMA (AT) 1990-06-06 CN disclosed
EP-0103553-B1 INTERMEDIATES FOR THE PREPARATION OF OMEPRAZOLE Aktiebolaget Hässle (SE) 1989-02-22 EP disclosed
US-4620008-A Processes for the preparation of omeprazole and intermediates therefore AKTIEBOLAGET HASSLE (SE) 1986-10-28 US disclosed
US-4544750-A Certain pyridyl-N-oxide intermediates for the preparation of omeprazole AKTIEBOLAGET HASSLE (SE) 1985-10-01 US disclosed
EP-0103553-A1 Intermediates for the preparation of omeprazole Aktiebolaget Hässle (SE) 1984-03-21 EP disclosed