SCHEMBL7952301

SCHEMBL7952301

COC(=O)C1=Nc2c(O)cc3c(c2C1)CC(O)CN3C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.34
USP30 Q70CQ3 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30
KDM1A O60341 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7945637 0.89 UCHL1 (0.34) UCHL1USP30HDAC1HDAC6
SCHEMBL7952298 0.74 UCHL1 (0.34) UCHL1USP30HDAC1HDAC6CYP1A2
SCHEMBL16568925 0.72 ADH1A (0.40) USP30HDAC1HDAC6CYP1A2POLB
SCHEMBL16569047 0.72 ADH1A (0.40) USP30HDAC1HDAC6CYP1A2POLB
SCHEMBL18406671 0.68 CYP1A2 (0.35) CYP1A2POLBCYP3A4CYP2C19CHRM2
SCHEMBL7945633 0.63 UCHL1 (0.34) UCHL1USP30HDAC1HDAC6
SCHEMBL14587286 0.62 KDM1A (0.46) HDAC1HDAC6CHRM2CHRM1CHRM3
SCHEMBL12268235 0.62 ALDH1A1 (0.48) UCHL1HDAC1HDAC6CHRM2CHRM1
SCHEMBL3738809 0.61 CHRM2 (0.53) CYP1A2POLBCYP3A4CYP2C19CHRM2
SCHEMBL18878053 0.61 CHRM2 (0.53) CYP1A2POLBCYP3A4CYP2C19CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281354-B1 ANTIBIOTICS; ANTITUMOR AGENTS THE SCRIPPS RESEARCH INSTITUTE 2001-08-28 US disclosed