SCHEMBL7952665

SCHEMBL7952665

O=S(=O)(Oc1ccc(OS(=O)(=O)C(F)(F)F)nc1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CXCR2 P25025 2/20 0.37
CXCR1 P25024 1/20 0.36
PDE4A P27815 3/20 0.36
PDE4C Q08493 3/20 0.36
PDE4D Q08499 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HTR1D P28221 3/20 0.35
HTR1A P08908 2/20 0.35
HTR1B P28222 2/20 0.35
CA9 Q16790 1/20 0.34
PTPRZ1 P23471 1/20 0.34
DRD2 P14416 2/20 0.34
DRD3 P35462 2/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RAB9A P51151 1/20 0.34
HSD11B1 P28845 1/20 0.34
PTPN1 P18031 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16559590 0.90 NFE2L2 (0.40) CA1CA2CXCR2CXCR1CA9
SCHEMBL22444656 0.88 SLC22A12 (0.43) CA1CA2CXCR2CXCR1MAPT
SCHEMBL30832531 0.84 CXCR2 (0.36) CA1CA2CXCR2PDE4APDE4C
SCHEMBL6852624 0.83 CA1 (0.40) CA1CA2CXCR2CXCR1HTR1D
SCHEMBL1017950 0.82 PDE4A (0.42) CA1CA2PDE4APDE4CPDE4D
SCHEMBL16548489 0.82 KDM4E (0.40) PDE4APDE4CPDE4DL3MBTL1MAPT
SCHEMBL3574836 0.82 ALDH1A1 (0.38) CA1CA2PDE4APDE4CPDE4D
SCHEMBL752015 0.80 CXCR2 (0.39) CA1CA2CXCR2CXCR1HTR1D
SCHEMBL1018963 0.80 PDE4A (0.41) CA1CA2PDE4APDE4CPDE4D
SCHEMBL8178203 0.80 L3MBTL1 (0.60) L3MBTL1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6262268-B1 REACTING 2,5-DI(3-PROPYLAMINO)PYRIDINE WITH BASE IN SOLVENT TO FORM 3-(5,6,7,8-TETRAHYDRO-(1,8)-NAPHTHYRIDIN-2-YL)-PROPYLAMINE AND ISOLATING PRODUCT MERCK & CO., INC. 2001-07-17 US disclosed