SCHEMBL7952836

SCHEMBL7952836

O=C(O)Cc1nc(=O)[nH]c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.53
ALDH1A1 P00352 5/20 0.53
HPGD P15428 3/20 0.53
HSD17B10 Q99714 2/20 0.53
TSHR P16473 1/20 0.53
ADORA3 P0DMS8 3/20 0.51
MAPT P10636 4/20 0.50
GAA P10253 2/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
LMNA P02545 1/20 0.50
APP P05067 2/20 0.49
EGFR P00533 2/20 0.49
AKR1B1 P15121 1/20 0.47
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11333762 0.81 KDM4E (0.56) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL26611803 0.79 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL31436766 0.79 APP (0.57) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL6191956 0.78 KDM4E (0.53) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL16914813 0.78 KDM4E (0.53) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL28337285 0.75 RAB9A (0.54) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL28847978 0.75 HPGD (0.43) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL29651055 0.75 LMNA (0.68) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL462088 0.75 LMNA (0.68) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL14072437 0.75 ADORA3 (0.68) KDM4EALDH1A1HPGDHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6258815-B1 HETEROCYCLIC COMPOUNDS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 2001-07-10 US claimed
US-6258815-B1 HETEROCYCLIC COMPOUNDS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 2001-07-10 US disclosed
US-4288362-A Monoazo pigments containing a quinazo linonylacetoacetanilide coupling component BAYER AKTIENGESELLSCHAFT (DE) 1981-09-08 US disclosed