SCHEMBL7953252

SCHEMBL7953252

CCn1ccc2c(OCCC(O)N3CCC(c4cccnc4)CC3)ccc(C(F)(F)F)c21

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.35
KCNH2 Q12809 5/20 0.35
GRM2 Q14416 1/20 0.34
CYP3A4 P08684 2/20 0.33
CCRL2 O00421 1/20 0.33
CTSS P25774 2/20 0.32
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HSD11B1 P28845 1/20 0.31
PDCD1LG2 Q9BQ51 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
PTK2 Q05397 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7953258 0.84 SLC18A3 (0.40) KCNH2
SCHEMBL7953261 0.82 GRM2 (0.35) CCR2KCNH2GRM2CCRL2CTSS
SCHEMBL7965925 0.74 HTR1A (0.47)
SCHEMBL13842724 0.62 CYP11B2 (0.57) TDP1
SCHEMBL16218244 0.62 CYP11B2 (0.57) KCNH2TDP1
SCHEMBL8871724 0.61 HTR1A (0.46)
SCHEMBL16755915 0.60 CYP11B2 (0.48) CCR2KCNH2GRM2TDP1HSD11B1
SCHEMBL12026531 0.60 CYP11B2 (0.50) TDP1HSD11B1
SCHEMBL23374726 0.58 CYP11B2 (0.53) CYP3A4TDP1
SCHEMBL4397664 0.58 CYP11B2 (0.62) CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
WO-2000006166-A1 5-HT1F ANTAGONISTS ELI LILLY AND COMPANY (US) 2000-02-10 WO disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed