SCHEMBL7953402

SCHEMBL7953402

CC(C)Sc1nc2c([nH]1)c(=O)n(Cc1ccc(Cl)cc1)c(=O)n2Cc1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
TSHR P16473 3/20 0.51
MAPK1 P28482 2/20 0.51
MAPT P10636 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
HPGD P15428 2/20 0.50
SIRT1 Q96EB6 5/20 0.46
SIRT3 Q9NTG7 5/20 0.46
SIRT5 Q9NXA8 5/20 0.46
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45
ADORA1 P30542 1/20 0.45
SIRT2 Q8IXJ6 1/20 0.45
TP53 P04637 2/20 0.44
XBP1 P17861 1/20 0.44
PKM P14618 1/20 0.43
HTT P42858 1/20 0.43
P2RX3 P56373 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7955637 0.94 SIRT1 (0.54) ALDH1A1TSHRMAPK1MAPTNPSR1
SCHEMBL3229725 0.82 ADORA2A (0.47) ADORA2AADORA2BADORA1P2RX3
SCHEMBL7091169 0.77 ADORA2B (0.48) ALDH1A1TSHRMAPK1HPGDSIRT1
SCHEMBL3111144 0.77 ADORA2B (0.48) ALDH1A1TSHRMAPK1HPGDSIRT1
SCHEMBL3231585 0.74 ADORA2A (0.57) ADORA2AADORA2BADORA1
SCHEMBL13940893 0.74 ADORA2B (0.60) ALDH1A1MEN1KMT2AADORA2AADORA2B
SCHEMBL7091342 0.71 KDM4E (0.42) ALDH1A1TSHRMAPK1MAPTNPSR1
SCHEMBL7953405 0.71 ADORA2A (0.41) ALDH1A1TSHRMAPK1MAPTNPSR1
SCHEMBL7424585 0.70 SIRT1 (0.58) TSHRMEN1KMT2ASIRT1SIRT3
SCHEMBL7091149 0.69 P2RX3 (0.41) ALDH1A1TSHRMAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6268373-B1 ENZYME INHIBITORS EURO-CELTIQUE S.A. (LU) 2001-07-31 US disclosed