SCHEMBL7954413

SCHEMBL7954413

CNc1ccccc1C(=O)NOCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.59
RAB9A P51151 8/20 0.59
PTGS2 P35354 2/20 0.59
ATM Q13315 2/20 0.50
KDM4E B2RXH2 2/20 0.50
POLB P06746 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.47
EGFR P00533 1/20 0.45
HDAC3 O15379 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7956547 0.84 RAB9A (0.68) NPC1RAB9APTGS2KDM4EKMT2A
SCHEMBL1715458 0.81 POLB (0.60) NPC1RAB9APTGS2POLBMEN1
SCHEMBL28681431 0.80 PTGS2 (0.64) NPC1RAB9APTGS2ATMKDM4E
SCHEMBL1715384 0.80 KDR (0.52) NPC1RAB9APTGS2KDM4EPOLB
SCHEMBL3636008 0.80 NPC1 (0.65) NPC1RAB9APTGS2KDM4EL3MBTL1
SCHEMBL28893760 0.80 NPC1 (0.65) NPC1RAB9APTGS2ATMKDM4E
SCHEMBL1714602 0.79 NPC1 (0.52) NPC1RAB9APTGS2ATMKDM4E
SCHEMBL1715854 0.79 KDM6B (0.53) NPC1RAB9APTGS2KDM4EPOLB
SCHEMBL24013287 0.78 ALDH1A1 (0.63) NPC1RAB9AATMKDM4EPOLB
SCHEMBL1715827 0.78 NPC1 (0.48) NPC1RAB9APTGS2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274383-B1 REACTING AN AMINO BOUND TO A SOLID SUPPORT WITH AN ISATOIC ANHYDRIDE TO FORM A 2-AMINOBENZAMIDE BOUND TO THE SUPPORT, AND THEN REACTING WITH ALDEHYDE USING A LEWIS ACID CATALYST TO FORM A 2,3-DIHYDRO-4(1H)-QUINAZOLINONE BOUND TO SUPPORT SEPRACOR INC. 2001-08-14 US disclosed