SCHEMBL7956031

SCHEMBL7956031

CCOC(=O)COc1cccc2cc(COCCOC(c3ccccc3)c3ccccc3)oc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2RL3 Q96RI0 2/20 0.43
ADORA2A P29274 3/20 0.40
ADORA3 P0DMS8 2/20 0.40
ADORA1 P30542 2/20 0.40
CASP3 P42574 1/20 0.39
CASP7 P55210 1/20 0.39
CASP9 P55211 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C19 P33261 2/20 0.39
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 1/20 0.38
ABCB1 P08183 1/20 0.37
HPGD P15428 2/20 0.37
CYP2D6 P10635 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958318 0.88 PTGIR (0.43) ADORA2AADORA3ADORA1CYP1A2CYP3A4
SCHEMBL7956745 0.83 PTGIR (0.47) ADORA2AADORA3ADORA1CYP1A2CYP3A4
SCHEMBL7958975 0.79 KDM4E (0.46) ADORA2AADORA3ADORA1CYP1A2CYP3A4
SCHEMBL7956033 0.78 F2RL3 (0.43) F2RL3ADORA2AADORA3ADORA1CASP3
SCHEMBL7956256 0.76 PTGIR (0.45) ADORA2AADORA3ADORA1CYP1A2CYP3A4
SCHEMBL7948818 0.74 KDM4E (0.45) ADORA2AADORA3ADORA1CYP1A2CYP3A4
SCHEMBL10933439 0.72 F2RL3 (0.56) F2RL3ADORA2AADORA3ADORA1CYP1A2
SCHEMBL10652147 0.71 LMNA (0.61) F2RL3ADORA2AADORA3ADORA1CYP1A2
SCHEMBL7956320 0.71 NPC1 (0.47) ADORA2AALDH1A1KDM4EHPGDPOLB
SCHEMBL10649757 0.70 F2RL3 (0.54) F2RL3ADORA2AADORA3ADORA1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6323235-B1 CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS AND ENZYME INHIBITORS OHTAKE ATSUSHI (JP) 2001-11-27 US disclosed
US-6043264-A A THROMBOXANE A2 RECEPTOR ANTAGONIST FOR TREATING HYPERTENSION, THROMBOSIS, ISCHEMIC HEART DISEASES, CIRCULATORY DISEASES, ARTERIOSCLEROSIS, PLATELET FUNCTION DISORDER, HYPERLIPIDEMIA, NEPHRITIS OR ASTHMA TORAY INDUSTRIES, INC. (JP) 2000-03-28 US disclosed
EP-0751126-A1 BENZENE-FUSED HETEROCYCLIC DERIVATIVE AND USE OF THE SAME TORAY INDUSTRIES, INC. (JP) 1997-01-02 EP disclosed