SCHEMBL7956733

SCHEMBL7956733

CC(C)Oc1ccc2c(c1)C(=O)CC(c1ccc3c(c1)OCO3)O2

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.67
NPC1 O15118 1/20 0.67
KMT2A Q03164 1/20 0.58
EDNRB P24530 1/20 0.56
EDNRA P25101 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27980886 0.79 RAB9A (0.61) RAB9ANPC1KMT2A
SCHEMBL27934733 0.78 MAOB (0.59) RAB9ANPC1KMT2A
SCHEMBL14759253 0.77 AR (0.52) RAB9ANPC1KMT2A
SCHEMBL7954475 0.76 EDNRB (0.71) EDNRBEDNRA
SCHEMBL27499329 0.75 KDM4E (0.56) RAB9AKMT2A
SCHEMBL7943851 0.75 EDNRB (0.76) EDNRBEDNRA
SCHEMBL7951769 0.75 EDNRB (0.54) EDNRBEDNRA
SCHEMBL7943804 0.75 EDNRB (0.87) EDNRBEDNRA
SCHEMBL27499330 0.75 EDNRB (0.55) EDNRB
SCHEMBL12341996 0.74 LMNA (0.52) RAB9ANPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103271904-B Nitric oxide donor endothelin receptor antagonist as well as preparation method and application thereof UNIV SOUTHEAST 2014-11-12 CN disclosed
CN-103271904-A Nitric oxide donor endothelin receptor antagonist as well as preparation method and application thereof UNIV SOUTHEAST 2013-09-04 CN disclosed
US-6218427-B1 AS ENDOTHELIN RECEPTOR ANTAGONIST SHIONOGI & CO., LTD. (JP) 2001-04-17 US disclosed
EP-0924207-A1 CHROMENE-3-CARBOXYLATE DERIVATIVES SHIONOGI & CO., LTD. (JP) 1999-06-23 EP disclosed