SCHEMBL7957271

SCHEMBL7957271

CCn1ncc2c(N[C@H](C)C3CCCCC3)c(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)cnc21

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 3/20 0.48
PDE4B Q07343 5/20 0.48
PDE4D Q08499 11/20 0.47
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7957275 1.00 IRAK4 (0.48) IRAK4PDE4BPDE4DALDH1A1HTT
SCHEMBL4492103 0.89 PDE4B (0.59) PDE4BPDE4D
SCHEMBL7955469 0.88 L3MBTL1 (0.49) IRAK4PDE4BPDE4D
SCHEMBL7955464 0.88 L3MBTL1 (0.49) IRAK4PDE4BPDE4D
SCHEMBL7956937 0.85 PDE4B (0.50) IRAK4PDE4BPDE4D
SCHEMBL7956928 0.85 PDE4B (0.50) IRAK4PDE4BPDE4D
SCHEMBL7959058 0.84 PDE5A (0.53) PDE4BPDE4D
SCHEMBL7959060 0.84 PDE5A (0.53) PDE4BPDE4D
SCHEMBL4345597 0.83 PDE4B (0.67) PDE4BPDE4D
SCHEMBL7955130 0.83 PDE4B (0.55) PDE4BPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326379-B1 ERECTILE DYSFUNCTION; CARDIOVASCULAR DISORDERS BRISTOL-MYERS SQUIBB CO. 2001-12-04 US disclosed