SCHEMBL7958731

SCHEMBL7958731

CN(C=O)/C(N)=N\C1CC(c2ccc(F)cc2)Oc2ccc(-c3cccc(C#N)c3)cc21

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 3/20 0.37
PAX8 Q06710 3/20 0.34
MCHR1 Q99705 1/20 0.33
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
KDM1A O60341 2/20 0.32
DPP4 P27487 2/20 0.31
DPP9 Q86TI2 2/20 0.31
DPP7 Q9UHL4 2/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
CTSD P07339 1/20 0.31
BACE1 P56817 1/20 0.31
NPY5R Q15761 1/20 0.31
DPP8 Q6V1X1 1/20 0.30
GPR88 Q9GZN0 1/20 0.30
HDAC2 Q92769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12299575 0.93 GPR88 (0.36) PAX8KDM1ADPP4DPP9DPP7
SCHEMBL7962464 0.85 BACE1 (0.33) CTSDBACE1
SCHEMBL882888 0.73 BACE1 (0.43) PAX8MCHR1DPP4DPP9DPP7
SCHEMBL7960735 0.73 CYP19A1 (0.34) MAOB
SCHEMBL7891697 0.69 BACE1 (0.38) CTSDBACE1
SCHEMBL12827653 0.68 BACE1 (0.40) DPP4DPP9DPP7BACE1DPP8
SCHEMBL882560 0.67 BACE1 (0.37) BACE1
SCHEMBL7961574 0.63 GPR88 (0.38) PAX8MCHR1KDM1AMAOAMAOB
SCHEMBL7958664 0.62 AR (0.31)
SCHEMBL7960933 0.62 CFTR (0.34) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110218192-A1 Inhibitors Of Beta-Secretase VITAE PHARMACEUTICALS, INC. (US) 2011-09-08 US disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110218192-A1 Inhibitors Of Beta-Secretase BACE1, BACE2, APP FADS1 1990/4885PAX8 4868/4885MCHR1 4797/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.