SCHEMBL7961574

SCHEMBL7961574

N#Cc1cccc(-c2ccc3c(c2)C(C(=O)N(Cc2ccccc2)C(=N)N)C[C@H](c2ccccc2)O3)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 2/20 0.38
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
FFAR2 O15552 1/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
ABCB1 P08183 2/20 0.34
MMP12 P39900 1/20 0.33
MMP13 P45452 1/20 0.33
XDH P47989 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
MCHR1 Q99705 1/20 0.33
KDM1A O60341 2/20 0.32
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
PAX8 Q06710 1/20 0.32
CFD P00746 1/20 0.32
F11 P03951 1/20 0.32
KLKB1 P03952 1/20 0.32
SCD O00767 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12299575 0.70 GPR88 (0.36) GPR88FFAR2CYP3A4XDHSLC22A12
SCHEMBL16136563 0.64 GPR88 (0.35) GPR88XDHSLC22A12CFDF11
SCHEMBL1822439 0.62 CYP19A1 (0.43) ABCB1XDHSLC22A12MAOAMAOB
SCHEMBL12300257 0.60 BACE1 (0.38)
SCHEMBL12244991 0.59 PGR (0.41)
SCHEMBL24328065 0.58 LMNA (0.60) DCUN1D1
SCHEMBL3058586 0.58 GRIN2D (0.51)
SCHEMBL3690613 0.57 GRIN2D (0.58)
SCHEMBL28768129 0.57 XDH (0.40) FFAR2XDHSLC22A12MCHR1PAX8
Hydrochloric Acid SCHEMBL27527274 0.57 GRIN2D (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed