SCHEMBL7964322

SCHEMBL7964322

O=C(Nc1ncccn1)C1=C(O)CCc2c1nc1ccccn21

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 5/20 0.43
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
PKM P14618 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPT P10636 2/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 2/20 0.39
CDK4 P11802 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
RAB9A P51151 2/20 0.38
PTGS2 P35354 1/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7961368 0.91 NTRK1 (0.39) NTRK1ALDH1A1KDM4EHPGDPKM
SCHEMBL7418872 0.89 NPC1 (0.42) NTRK1ALDH1A1KDM4EPKMKMT2A
SCHEMBL7418952 0.86 RAB9A (0.44) NTRK1KMT2ARAB9ANPC1GAA
SCHEMBL7958240 0.85 IKBKE (0.41) NTRK1KDM4EMAPTKMT2ARAB9A
SCHEMBL7964125 0.85 NTRK1 (0.43) NTRK1ALDH1A1KDM4EHPGDPOLB
SCHEMBL7420479 0.85 NTRK1 (0.43) NTRK1ALDH1A1KDM4EMAPTPOLB
SCHEMBL8873046 0.85 CHRNB2 (0.41) NTRK1ALDH1A1KDM4EHPGDPKM
SCHEMBL7960418 0.85 NTRK1 (0.37) NTRK1ALDH1A1KDM4EHPGDPKM
SCHEMBL7959855 0.84 LMNA (0.44) NTRK1HPGDMAPTPOLBKMT2A
SCHEMBL7964540 0.84 NPC1 (0.51) ALDH1A1KDM4EHPGDPKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US claimed
US-6218384-B1 FOR THERAPY OF ANXIETY, MUSCLE SPASMS, SLEEPLESSNESS, CONVULSIONS AND BENZODIAZEPINE OVERDOSES ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-04-17 US disclosed
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US disclosed