SCHEMBL7960425

SCHEMBL7960425

Cc1ccc2c(c1)N(CC(=O)c1cccs1)C(=O)C(NC(=O)OC(C)(C)C)CN2C(=O)c1cccs1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
TSHR P16473 1/20 0.40
CCKBR P32239 3/20 0.37
MAPK1 P28482 1/20 0.36
TP53 P04637 2/20 0.36
MAPT P10636 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HTT P42858 1/20 0.35
SCN9A Q15858 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7962064 0.93 CCKBR (0.36) ALDH1A1TSHRCCKBRTP53MAPT
SCHEMBL6177954 0.92 TP53 (0.38) ALDH1A1TSHRCCKBRMAPK1TP53
SCHEMBL6177683 0.91 CCKBR (0.36) ALDH1A1TSHRCCKBRTP53CYP1A2
SCHEMBL6180722 0.81 ALDH1A1 (0.47) ALDH1A1TSHRMAPK1TP53MAPT
SCHEMBL6176477 0.80 MEN1 (0.40) ALDH1A1TSHRCCKBRMAPK1TP53
SCHEMBL6178050 0.80 CCKBR (0.50) CCKBR
SCHEMBL7959374 0.80 ALDH1A1 (0.43) ALDH1A1TSHRMAPK1TP53MAPT
SCHEMBL6177504 0.80 CCKBR (0.39) TSHRCCKBRMAPT
SCHEMBL6176679 0.79 CCKBR (0.46) TSHRCCKBRMAPT
SCHEMBL6177392 0.78 CCKBR (0.39) TSHRCCKBRMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed