SCHEMBL7962064

SCHEMBL7962064

Cc1ccc2c(c1)N(CC(=O)c1cccs1)C(=O)C(NC(=O)OC(C)(C)C)CN2C(=O)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 3/20 0.36
ALDH1A1 P00352 4/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
SCN9A Q15858 5/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
TSHR P16473 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7960425 0.93 ALDH1A1 (0.40) CCKBRALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL6177683 0.91 CCKBR (0.36) CCKBRALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL7960830 0.85 CCKBR (0.35) CCKBRSCN9ALMNATSHR
SCHEMBL6177954 0.85 TP53 (0.38) CCKBRALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL6176603 0.85 CCKBR (0.39) CCKBRSCN9ALMNATSHRMAPT
SCHEMBL6181983 0.84 CCKBR (0.36) CCKBRALDH1A1SCN9ALMNATP53
SCHEMBL6178413 0.83 ALDH1A1 (0.40) ALDH1A1CYP1A2CYP2D6CYP2C19LMNA
SCHEMBL7959681 0.83 CCKBR (0.35) CCKBRSCN9A
SCHEMBL6176746 0.82 CCKBR (0.52) CCKBR
SCHEMBL6177998 0.82 CCKBR (0.47) CCKBRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed