SCHEMBL6180722

SCHEMBL6180722

Cc1ccc2c(c1)N(CC(=O)c1cccs1)C(=O)C(N)CN2C(=O)c1cccs1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 2/20 0.38
HTT P42858 1/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
PABPC1 P11940 1/20 0.37
APOBEC3A P31941 1/20 0.37
EIF4H Q15056 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
KCNA5 P22460 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6176322 0.91 TSHR (0.43) ALDH1A1TSHRMAPK1CYP1A2CYP2D6
SCHEMBL6178413 0.90 ALDH1A1 (0.40) ALDH1A1TSHRMAPK1CYP1A2CYP2D6
SCHEMBL6175739 0.88 ALDH1A1 (0.39) ALDH1A1TSHRMAPK1CYP1A2CYP2D6
SCHEMBL7960425 0.81 ALDH1A1 (0.40) ALDH1A1TSHRMAPK1CYP1A2CYP2D6
SCHEMBL6178050 0.77 CCKBR (0.50)
SCHEMBL6176477 0.76 MEN1 (0.40) ALDH1A1TSHRMAPK1CYP1A2CYP2D6
SCHEMBL6176470 0.74 TSHR (0.42) ALDH1A1TSHRMAPK1CYP1A2CYP2D6
SCHEMBL6177954 0.74 TP53 (0.38) ALDH1A1TSHRMAPK1CYP1A2CYP2D6
SCHEMBL7962064 0.73 CCKBR (0.36) ALDH1A1TSHRCYP1A2CYP2D6CYP2C19
SCHEMBL6209886 0.72 TSHR (0.35) ALDH1A1TSHRCYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945445-B9 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2005-12-28 EP disclosed
EP-0945445-B1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2003-09-03 EP disclosed
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed
EP-0945445-A1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed