SCHEMBL7963355

SCHEMBL7963355

C=CCONC(=O)c1ccccc1N

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.62
HSD17B10 Q99714 5/20 0.62
TSHR P16473 1/20 0.62
CYP3A4 P08684 1/20 0.49
LIG1 P18858 1/20 0.48
CFTR P13569 1/20 0.46
KDM4E B2RXH2 9/20 0.43
HPGD P15428 7/20 0.43
RCE1 Q9Y256 1/20 0.43
FADS1 O60427 1/20 0.42
TP53 P04637 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
USP2 O75604 1/20 0.41
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30012222 0.84 CA1 (0.50) ALDH1A1HSD17B10TSHRCYP3A4LIG1
SCHEMBL29035769 0.83 CA1 (0.49) ALDH1A1HSD17B10TSHRCYP3A4LIG1
SCHEMBL31247461 0.83 CA1 (0.49) ALDH1A1HSD17B10TSHRCYP3A4LIG1
SCHEMBL1558090 0.78 ALDH1A1 (0.59) ALDH1A1HSD17B10TSHRCFTRKDM4E
SCHEMBL5318792 0.78 NPC1 (0.59) ALDH1A1HSD17B10CYP3A4LIG1HPGD
SCHEMBL143432 0.77 ALDH1A1 (0.49) ALDH1A1HSD17B10TSHRCYP3A4CFTR
SCHEMBL10785014 0.77 ALDH1A1 (0.49) ALDH1A1HSD17B10TSHRCYP3A4CFTR
SCHEMBL759012 0.77 ALDH1A1 (1.00) ALDH1A1HSD17B10TSHRCYP3A4LIG1
SCHEMBL1561753 0.77 HPGD (0.66) ALDH1A1HSD17B10TSHRCYP3A4KDM4E
SCHEMBL3636008 0.75 NPC1 (0.65) ALDH1A1HSD17B10TSHRCYP3A4CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274383-B1 REACTING AN AMINO BOUND TO A SOLID SUPPORT WITH AN ISATOIC ANHYDRIDE TO FORM A 2-AMINOBENZAMIDE BOUND TO THE SUPPORT, AND THEN REACTING WITH ALDEHYDE USING A LEWIS ACID CATALYST TO FORM A 2,3-DIHYDRO-4(1H)-QUINAZOLINONE BOUND TO SUPPORT SEPRACOR INC. 2001-08-14 US claimed