SCHEMBL7963988

SCHEMBL7963988

CC(C)(C)OC(=O)N(CCCNc1cccc(-c2cccnc2C(=O)Nc2ccccc2)c1)C[C@@H](O[Si](C)(C)C(C)(C)C)c1cccc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.37
NPSR1 Q6W5P4 5/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPK1 P28482 2/20 0.37
ADRB1 P08588 6/20 0.34
ADRB3 P13945 6/20 0.34
GRM4 Q14833 1/20 0.34
ADRB2 P07550 5/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
BACE1 P56817 1/20 0.34
TDP1 Q9NUW8 3/20 0.33
ATR Q13535 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
KLRK1 P26718 1/20 0.33
MICA Q29983 1/20 0.33
RAET1L Q5VY80 1/20 0.33
IDO1 P14902 1/20 0.33
TRPV4 Q9HBA0 1/20 0.32
NTSR1 P30989 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7975406 0.96 MAPT (0.38) MAPTNPSR1KDM4EMAPK1ADRB1
SCHEMBL7975401 0.96 MAPT (0.38) MAPTNPSR1KDM4EMAPK1ADRB1
SCHEMBL7963984 0.86 ADRB1 (0.39) MAPTNPSR1KDM4EMAPK1ADRB1
SCHEMBL7963987 0.86 ADRB1 (0.39) MAPTNPSR1KDM4EMAPK1ADRB1
SCHEMBL6433084 0.84 ADRB1 (0.42) ADRB1ADRB3ADRB2SMN1; SMN2BACE1
SCHEMBL7964117 0.82 ADRB1 (0.46) ADRB1ADRB3ADRB2KLRK1MICA
SCHEMBL7975458 0.80 ADRB2 (0.44) ADRB1ADRB3ADRB2
SCHEMBL5949915 0.79 ADRB1 (0.43) MAPTNPSR1KDM4EMAPK1ADRB1
SCHEMBL5950125 0.79 ADRB1 (0.44) ADRB1ADRB3ADRB2
SCHEMBL6436894 0.79 ADRB1 (0.44) ADRB1ADRB3ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001042217-A1 BETA-3 ADRENOCEPTOR AGONISTS GLAXO GROUP LIMITED (GB) 2001-06-14 WO disclosed