SCHEMBL796459

SCHEMBL796459

CC(=O)c1ccc(-c2nc(-c3nc(N)nc(N(C)c4ccccc4)n3)no2)nc1.CC(O)c1ccc(-c2nc(-c3nc(N)nc(N(C)c4ccccc4)n3)no2)nc1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.33
HCAR2 Q8TDS4 3/20 0.33
TPH1 P17752 1/20 0.33
ATR Q13535 3/20 0.32
HDAC1 Q13547 2/20 0.32
S1PR1 P21453 2/20 0.31
S1PR3 Q99500 1/20 0.31
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL796822 0.93 HCAR2 (0.33) HDAC4HCAR2TPH1ATRS1PR1
SCHEMBL795346 0.92 ATR (0.36) HDAC4HCAR2ATRHDAC1HDAC6
SCHEMBL795809 0.82 MAPT (0.36) ATRHDAC1HDAC6
SCHEMBL15480817 0.80 DHFR (0.36) ATR
SCHEMBL797169 0.79 NPC1 (0.33)
SCHEMBL796527 0.78 GRM5 (0.38) HCAR2
SCHEMBL795257 0.77 HDAC4 (0.35) HDAC4HDAC1S1PR1S1PR3HDAC6
SCHEMBL794849 0.77 GABRA5 (0.42) HDAC4HDAC1HDAC6
SCHEMBL796056 0.77 NPC1 (0.41) S1PR1
SCHEMBL796460 0.77 ATR (0.34) HDAC4ATRHDAC1S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150025057-A1 Triazine-oxadiazoles NOVARTIS AG (CH) 2015-01-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150025057-A1 Triazine-oxadiazoles OPRK1, OPRD1, OPRL1 HDAC4 781/4885HCAR2 643/4885TPH1 154/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.