SCHEMBL7965283

SCHEMBL7965283

C[C](C)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.55
TYR P14679 1/20 0.55
HDAC1 Q13547 1/20 0.54
SRD5A2 P31213 1/20 0.52
TSHR P16473 1/20 0.50
MAPT P10636 3/20 0.47
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HTT P42858 2/20 0.47
KMT2A Q03164 2/20 0.47
HIF1A Q16665 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
POLB P06746 1/20 0.47
RARB P10826 1/20 0.47
RARG P13631 1/20 0.47
SIRT1 Q96EB6 1/20 0.45
EPHX2 P34913 2/20 0.44
NR1H4 Q96RI1 2/20 0.44
ALOX12 P18054 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL292571 0.80 LMNA (0.57) LMNATYRHDAC1SRD5A2TSHR
SCHEMBL465848 0.79 TSHR (0.52) LMNATYRHDAC1SRD5A2TSHR
SCHEMBL11699186 0.79 MAPT (0.50) LMNATYRHDAC1SRD5A2TSHR
SCHEMBL397829 0.79 EPHX2 (0.65) LMNATYRHDAC1SRD5A2MAPT
SCHEMBL9889072 0.79 HDAC1 (0.50) LMNATYRHDAC1SRD5A2TSHR
SCHEMBL424728 0.78 TSHR (0.73) LMNATYRHDAC1SRD5A2TSHR
SCHEMBL1552000 0.78 ESR1 (0.38) LMNATSHRMAPTMEN1ALDH1A1
SCHEMBL14471516 0.78 SRD5A2 (0.58) LMNATYRHDAC1SRD5A2TSHR
SCHEMBL22363237 0.77 HDAC1 (0.48) LMNATYRHDAC1SRD5A2TSHR
SCHEMBL22363236 0.77 HDAC1 (0.48) LMNATYRHDAC1SRD5A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023101004-A1 OLEFIN RESIN, METHOD FOR MANUFACTURING SAME, AND APPLICATION FOR SAME 三井化学株式会社 2023-06-08 WO disclosed
US-6291472-B1 4a, 5a, 8a, 8b-tetrahydro-6H-pyrrolo[3′,4′:4, 5]furo[3,2-b] pyri-dine-6,8(7H)-dione derivatives for control of endoparasites processes for their preparation BAYER AKTIENGESELLSCHAFT (DE) 2001-09-18 US disclosed
US-6110928-A HUMAN OR VETERINARY MEDICINE BAYER AKTIENGESELLSCHAFT (DE) 2000-08-29 US disclosed
EP-0377633-B1 PEROXIDE FREE RADICAL INITIATORS CONTAINING HINDERED AMINE LIGHT STABILIZER GROUPS ATOCHEM NORTH AMERICA (US) 1995-05-17 EP disclosed
US-5234946-A Anticholesterol, antilipemic BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-10 US disclosed
EP-0318860-B1 SUBSTITUTED ALKYLAMINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-16 EP disclosed
EP-0377633-A4 PEROXIDE FREE RADICAL INITIATORS CONTAINING HINDERED AMINE LIGHT STABILIZER GROUPS 1991-01-30 EP disclosed
EP-0377633-A1 PEROXIDE FREE RADICAL INITIATORS CONTAINING HINDERED AMINE LIGHT STABILIZER GROUPS. PENNWALT CORP (US) 1990-07-18 EP disclosed
US-4925903-A PEROXIDE CONTAINING HINDERED AMINE ALSO FUNCTIONS AS INITIATOR PENNWALT CORPORATION (US) 1990-05-15 US disclosed
US-4885347-A UNSATURATED POLYESTER PENNWALT CORPORATION (US) 1989-12-05 US disclosed
EP-0318860-A2 Substituted alkylamine derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1989-06-07 EP disclosed
US-4822883-A 2,2,6,6-TETRA SUBSTITUTED PIPERIDIN-4-YL PEROXY DERIVATIVES BECOMING CHEMICALLY BONDED TO ADDITION POLYMER PENNWALT CORPORATION (US) 1989-04-18 US disclosed
WO-1989001474-A1 PEROXIDE FREE RADICAL INITIATORS CONTAINING HINDERED AMINE LIGHT STABILIZER GROUPS PENNWALT CORPORATION (US) 1989-02-23 WO disclosed