SCHEMBL465848

SCHEMBL465848

C=C(C)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
HDAC1 Q13547 1/20 0.50
LMNA P02545 1/20 0.50
TYR P14679 1/20 0.50
MAPT P10636 3/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
SRD5A2 P31213 1/20 0.48
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HTT P42858 2/20 0.44
KMT2A Q03164 2/20 0.44
HIF1A Q16665 1/20 0.44
POLB P06746 1/20 0.44
RARB P10826 1/20 0.44
RARG P13631 1/20 0.44
SIRT1 Q96EB6 1/20 0.42
EPHX2 P34913 2/20 0.42
NR1H4 Q96RI1 2/20 0.42
ALOX12 P18054 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9017221 0.91 L3MBTL1 (0.49) TSHRHDAC1LMNATYRMAPT
SCHEMBL11281234 0.85 ESR1 (0.43) TSHRHDAC1LMNATYRMAPT
SCHEMBL13889245 0.84 NPC1 (0.53) TSHRHDAC1LMNAMAPTNPC1
SCHEMBL13987317 0.83 MAPT (0.42) TSHRHDAC1LMNATYRMAPT
SCHEMBL6563424 0.83 TSHR (0.37) TSHRHDAC1LMNATYRMAPT
SCHEMBL28160104 0.82 LMNA (0.52) TSHRHDAC1LMNATYRMAPT
SCHEMBL13747948 0.82 RAB9A (0.41) TSHRLMNAMAPTNPC1RAB9A
SCHEMBL8677283 0.81 TSHR (0.36) TSHRHDAC1LMNATYRMAPT
SCHEMBL11116753 0.81 TSHR (0.36) TSHRHDAC1LMNATYRMAPT
SCHEMBL7253138 0.81 PDE2A (0.43) TSHRHDAC1LMNAMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 298 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2345679-B1 METHOD FOR PRODUCING GRAFT COPOLYMER, GRAFT COPOLYMER OBTAINED BY THE METHOD, RUBBER COMPOSITION CONTAINING THE GRAFT COPOLYMER, AND TIRE BRIDGESTONE CORP (JP) 2016-04-27 EP claimed
US-8722806-B2 Rubber composition and tire using the same BRIDGESTONE CORPORATION (JP) 2014-05-13 US claimed
EP-2248851-B1 RUBBER COMPOSITION AND TIRE USING THE SAME BRIDGESTONE CORP (JP) 2013-05-29 EP claimed
US-20110224351-A1 METHOD FOR PRODUCING GRAFT COPOLYMER, GRAFT COPOLYMER OBTAINED BY THE METHOD, RUBBER COMPOSITION CONTAINING THE GRAFT COPOLYMER, AND TIRE BRIDGESTONE CORPORATION (JP) 2011-09-15 US claimed
US-20110196100-A1 RUBBER COMPOSITION AND TIRE USING THE SAME BRIDGESTONE CORPORATION (JP) 2011-08-11 US claimed
EP-2345679-A1 METHOD FOR PRODUCING GRAFT COPOLYMER, GRAFT COPOLYMER OBTAINED BY THE METHOD, RUBBER COMPOSITION CONTAINING THE GRAFT COPOLYMER, AND TIRE Bridgestone Corporation (JP) 2011-07-20 EP claimed
EP-2248851-A1 RUBBER COMPOSITION AND TIRE USING THE SAME Bridgestone Corporation (JP) 2010-11-10 EP claimed
JP-4372014-B2 2009-11-25 JP claimed
JP-2006506415-A 2006-02-23 JP claimed
EP-1599487-A1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE Givaudan SA (CH) 2005-11-30 EP claimed
WO-2004048394-A1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE GIVAUDAN SA (CH) 2004-06-10 WO claimed
WO-2004043971-A1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE GIVAUDAN SA (CH) 2004-05-27 WO claimed
US-4839203-A COVALENT BONDING PRODUCING A COMPOSITE THE DOW CHEMICAL COMPANY (US) 1989-06-13 US claimed
US-4797187-A COACERVATION OF CATIONS THE DOW CHEMICAL COMPANY (US) 1989-01-10 US claimed
US-4709109-A Preparation of alkenylaromatics BASF AKTIENGESELLSCHAFT (DE) 1987-11-24 US claimed
US-4704324-A REVERSE OSMOSIS, GAS SEPARATION, ULTRAFILTRATION THE DOW CHEMICAL COMPANY (US) 1987-11-03 US claimed
EP-4508056-B1 INDOLE-FUNCTIONALIZED BISPHOSPHORAMIDITES, METHODS FOR THE PREPARATION THEREOF, AND RHODIUM-LIGAND COMPLEX DOW GLOBAL TECHNOLOGIES LLC (US) 2026-05-06 EP disclosed
EP-4608553-A1 HETEROGENEOUS CATALYSTS DOW GLOBAL TECHNOLOGIES LLC (US) 2025-09-03 EP disclosed
US-4156763-A ORGANOLITHIUM INITIATOR TO PRODUCE RANDOM POLYMER PHILLIPS PETROLEUM COMPANY (US) 1979-05-29 US disclosed
US-4133835-A REACTING AN OLEFIN, A HALIDE, AND A HYDROPEROXIDE PENNWALT CORPORATION (US) 1979-01-09 US disclosed