SCHEMBL7966071

SCHEMBL7966071

NC(=O)C1(O)CN(C2CCC(c3ccccn3)CC2)C1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.39
DRD2 P14416 4/20 0.39
DRD3 P35462 3/20 0.39
HSD11B1 P28845 1/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CCRL2 O00421 1/20 0.38
CCR2 P41597 1/20 0.38
KCNH2 Q12809 1/20 0.38
OPRM1 P35372 2/20 0.38
OPRL1 P41146 2/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7966073 0.82 TRPV6 (0.41) DRD4MAPTTDP1CCRL2CCR2
SCHEMBL7967371 0.81 CCRL2 (0.43) DRD4DRD2DRD3HSD11B1CCRL2
Hydrochloric Acid SCHEMBL7971160 0.80 CCRL2 (0.43) DRD4DRD2DRD3HSD11B1MAPT
Carbamic Acid SCHEMBL10474895 0.78 ALDH1A1 (0.46) DRD4DRD2DRD3HSD11B1MAPT
SCHEMBL30131210 0.74 KMT2A (0.47) DRD4DRD2DRD3HSD11B1MAPT
SCHEMBL16803154 0.74 KMT2A (0.47) DRD4DRD2DRD3HSD11B1MAPT
Hydrochloric Acid SCHEMBL30562858 0.73 KMT2A (0.46) DRD4DRD2DRD3HSD11B1MAPT
SCHEMBL900225 0.72
SCHEMBL659325 0.72 KDM4E (0.48) DRD4DRD2DRD3HSD11B1MAPT
SCHEMBL29448519 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255315-B1 BENIGN PROSTATIC HYPERPLASIA MERCK & CO., INC. 2001-07-03 US disclosed
US-6037354-A ADMINISTERING PHENYL-SUBSTITUTED THIAZOLIDIN-4-ONE OR OXAZOLIDIN-2-ONE DERIVATIVE TO TREAT BENIGN PROSTATE HYPERPLASIA; SIDE EFFECT REDUCTION MERCK & CO., INC. (US) 2000-03-14 US disclosed