SCHEMBL7966084

SCHEMBL7966084

CC(C)(C)OC(=O)NCCCN1CCC(C#N)(c2ccccc2)CC1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 6/20 0.66
ADRA1A P35348 6/20 0.66
ADRA1B P35368 5/20 0.66
DRD2 P14416 8/20 0.59
OPRM1 P35372 1/20 0.54
SIGMAR1 Q99720 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7670825 0.90 DRD2 (0.59) ADRA1DADRA1AADRA1BDRD2
SCHEMBL6961341 0.90 DRD2 (0.74) ADRA1DADRA1AADRA1BDRD2OPRM1
SCHEMBL7663181 0.90 DRD2 (0.59) ADRA1DADRA1AADRA1BDRD2
SCHEMBL7956108 0.87 ADRA1D (0.68) ADRA1DADRA1AADRA1BDRD2
SCHEMBL7702063 0.86 ADRA1A (0.55) ADRA1DADRA1AADRA1BDRD2
SCHEMBL7965434 0.86 ADRA1D (0.66) ADRA1DADRA1AADRA1BDRD2
SCHEMBL7566269 0.84 DRD2 (0.63) ADRA1DADRA1AADRA1BDRD2SIGMAR1
SCHEMBL14902481 0.83 SIGMAR1 (0.56) ADRA1DADRA1AADRA1BDRD2SIGMAR1
SCHEMBL14902477 0.82 SIGMAR1 (0.60) ADRA1DADRA1AADRA1BDRD2SIGMAR1
SCHEMBL7531578 0.81 ADRA1A (0.59) ADRA1DADRA1AADRA1BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274583-B1 Alpha 1a adrenergic receptor antagonists MERCK & CO., INC. 2001-08-14 US disclosed
US-5977115-A Alpha 1a adrenergic receptor antagonists MERCK & CO., INC. (US) 1999-11-02 US disclosed