SCHEMBL7966573

SCHEMBL7966573

CCC(CCC(C#N)(c1ccc(C(F)(F)F)cc1)C(C)C)N(C(C)c1ccccc1)C(C)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.41
EBP Q15125 2/20 0.41
SLC6A4 P31645 3/20 0.36
HRH3 Q9Y5N1 2/20 0.36
SLC6A9 P48067 4/20 0.35
AR P10275 4/20 0.34
CYP2D6 P10635 4/20 0.33
CYP2C19 P33261 3/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
LMNA P02545 3/20 0.33
NPC1 O15118 2/20 0.33
MTOR P42345 2/20 0.33
RAB9A P51151 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
TSHR P16473 2/20 0.33
SLC6A2 P23975 2/20 0.33
ACP3 P15309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968877 0.91 EBP (0.41) SIGMAR1EBPSLC6A4SLC6A9CYP2D6
SCHEMBL7965756 0.91 EBP (0.43) SIGMAR1EBPSLC6A4HRH3SLC6A9
SCHEMBL7965402 0.89 EBP (0.41) SIGMAR1EBPSLC6A4CYP2D6CYP2C19
SCHEMBL7968976 0.89 EBP (0.41) SIGMAR1EBPSLC6A4CYP2D6MEN1
SCHEMBL7971875 0.87 SIGMAR1 (0.43) SIGMAR1EBPSLC6A4HRH3SLC6A9
SCHEMBL7968875 0.83 SIGMAR1 (0.45) SIGMAR1EBPSLC6A4MEN1KMT2A
SCHEMBL7972074 0.82 SIGMAR1 (0.46) SIGMAR1EBPSLC6A4HRH3SLC6A9
SCHEMBL7969252 0.82 SIGMAR1 (0.47) SIGMAR1EBPSLC6A4CYP2D6CYP2C19
SCHEMBL7968647 0.82 EBP (0.43) SIGMAR1EBPSLC6A4SLC6A9AR
SCHEMBL7967345 0.81 SIGMAR1 (0.43) SIGMAR1EBPSLC6A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed