SCHEMBL7967090

SCHEMBL7967090

CC(CCC(C#N)(c1c(C(F)(F)F)cccc1C(F)(F)F)C(C)C)N(C)Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
ADRA1A P35348 2/20 0.41
OPRK1 P41145 2/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2A P28223 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KCNH2 Q12809 1/20 0.41
EBP Q15125 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
MAOB P27338 5/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
EPHX2 P34913 1/20 0.33
MAOA P21397 4/20 0.33
CYP1A2 P05177 2/20 0.33
ADRA2A P08913 1/20 0.33
SNCA P37840 1/20 0.33
CYP2D6 P10635 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968611 0.91 ADRA2B (0.43) ADRA2BADRA2CADRA1AOPRK1SLC6A2
SCHEMBL7969369 0.89 SIGMAR1 (0.48) ADRA2BADRA2CADRA1AHTR2ASLC6A4
SCHEMBL7971756 0.88 EBP (0.38) ADRA2BADRA2CADRA1AOPRK1SLC6A2
SCHEMBL7969852 0.88 EBP (0.37) SLC6A2SLC6A4EBPSIGMAR1L3MBTL1
SCHEMBL7967041 0.87 BCHE (0.39) ADRA2BSLC6A2HTR2ASLC6A4KCNH2
SCHEMBL7966372 0.86 ADRA2B (0.43) ADRA2BADRA2CADRA1AOPRK1SLC6A2
SCHEMBL7971694 0.85 BCHE (0.41) ADRA2BADRA2CADRA1AOPRK1SLC6A2
SCHEMBL7968778 0.84 ADRA2B (0.43) ADRA2BADRA2CADRA1AOPRK1SLC6A2
SCHEMBL7965566 0.84 ADRA2B (0.43) ADRA2BADRA2CADRA1AOPRK1SLC6A2
SCHEMBL7971844 0.84 ADRA2B (0.43) ADRA2BADRA2CADRA1AOPRK1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed