SCHEMBL7967262

SCHEMBL7967262

COc1ccc2cc(C3(O)CCN(C(=O)OC(C)(C)C)CC3)ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
BACE1 P56817 2/20 0.47
CTSD P07339 1/20 0.47
CTSE P14091 1/20 0.47
STS P08842 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
GPR119 Q8TDV5 1/20 0.45
EPHX2 P34913 1/20 0.43
HTT P42858 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802425 0.89 ALDH1A1 (0.55) ALDH1A1BACE1CTSDCTSESTS
Water SCHEMBL8370294 0.87 ALDH1A1 (0.40) ALDH1A1BACE1CTSDCTSESTS
SCHEMBL5240524 0.87 ALDH1A1 (0.65) ALDH1A1SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL16874679 0.84 ALDH1A1 (0.51) ALDH1A1BACE1CTSDCTSESTS
SCHEMBL8398896 0.83 YAP1 (0.49) GPR119
SCHEMBL15595077 0.83 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL5759621 0.82 KDM4E (0.41) ALDH1A1BACE1CTSDCTSESTS
SCHEMBL6159582 0.82 LMNA (0.49) ALDH1A1BACE1CTSDCTSESTS
SCHEMBL16874616 0.82 L3MBTL1 (0.50) ALDH1A1BACE1CTSDCTSESTS
SCHEMBL6311972 0.81 ALDH1A1 (0.46) ALDH1A1BACE1CTSDCTSESTS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303627-B1 FOR THERAPY OF PHYSIOLOGICAL AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY 2001-10-16 US disclosed
WO-1999065487-A1 INHIBITORS OF SEROTONIN REUPTAKE ELI LILLY AND COMPANY (US) 1999-12-23 WO disclosed
EP-0965587-A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1999-12-22 EP disclosed