SCHEMBL7967300

SCHEMBL7967300

CC(C)c1ccc2cnc(C3CCNCC3)cc2c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 9/20 0.43
TLR8 Q9NR97 9/20 0.43
TLR7 Q9NYK1 9/20 0.43
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
GSK3B P49841 2/20 0.38
DYRK1A Q13627 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
MAPK8 P45983 1/20 0.36
BRD4 O60885 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
MMP9 P14780 1/20 0.35
AKT1 P31749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7954797 0.79 TLR9 (0.44) TLR9TLR8TLR7SLC6A2SLC6A4
SCHEMBL5241881 0.77 BCHE (0.45) SLC6A2SLC6A4SLC6A3L3MBTL1HRH4
Hydrochloric Acid SCHEMBL3880186 0.76 BCHE (0.44) SLC6A2SLC6A4SLC6A3L3MBTL1HRH4
SCHEMBL24218862 0.73 GSK3B (0.64) GSK3BDYRK1A
SCHEMBL7955491 0.72 L3MBTL1 (0.40) TLR9TLR8TLR7SLC6A2SLC6A4
SCHEMBL10834084 0.72 HRH4 (0.46) SLC6A2SLC6A4L3MBTL1HRH4GABRA1
SCHEMBL10262259 0.69 CYP1A2 (0.53)
SCHEMBL10199297 0.69 GRM4 (0.42)
SCHEMBL7971282 0.69 RAB9A (0.64) TLR9TLR8TLR7SLC6A2SLC6A4
SCHEMBL18319496 0.68 DYRK1A (0.51) GSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303627-B1 FOR THERAPY OF PHYSIOLOGICAL AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY 2001-10-16 US disclosed
EP-0965587-A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1999-12-22 EP disclosed