SCHEMBL7967646

SCHEMBL7967646

O=C1CNCCN1Cc1cnc[nH]1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.46
HRH3 Q9Y5N1 10/20 0.40
HRH4 Q9H3N8 7/20 0.40
FNTA P49354 2/20 0.37
FNTB P49356 2/20 0.37
CYP2D6 P10635 1/20 0.37
PKM P14618 1/20 0.37
MPG P29372 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
GABRA1 P14867 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
GABRR1 P24046 1/20 0.37
GABRR2 P28476 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRB2 P47870 1/20 0.37
GABRA4 P48169 1/20 0.37
HRH1 P35367 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2337242 0.78 TAAR1 (0.59) TAAR1HRH3HRH4CYP2D6PKM
Trifluoroacetic Acid SCHEMBL7363253 0.74 HRH3 (0.55) HRH3HRH4HRH1
SCHEMBL27574319 0.74 DRD2 (0.41) CYP2D6ALDH1A1CYP3A4
SCHEMBL14993193 0.72 ALDH1A1 (0.53) ALDH1A1
SCHEMBL4397329 0.71 F10 (0.51) HRH4
Hydrochloric Acid SCHEMBL1306753 0.71 ALDH1A1 (0.52) ALDH1A1
SCHEMBL30282988 0.70 KDM4E (0.37) CYP2D6ALDH1A1CYP3A4TSHRNFKB1
SCHEMBL21133356 0.70 MPG (0.43) TAAR1HRH3HRH4FNTAFNTB
SCHEMBL92331 0.69 L3MBTL1 (0.56) CYP2D6ALDH1A1TSHR
SCHEMBL17525758 0.69 TAAR1 (0.46) TAAR1HRH3HRH4PKMMPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001007437-A1 CRYSTAL FORMS OF 1-(3-CHLOROPHENYL)-4-[1-(4-CYANOBENZYL)-5-IMIDAZOLYLMETHYL]-2-PIPERAZINONE MERCK & CO., INC. (US) 2001-02-01 WO disclosed
WO-2000001691-A1 PROCESS FOR MAKING FARNESYL-PROTEIN TRANSFERASE INHIBITORS MERCK & CO., INC. (US) 2000-01-13 WO disclosed