SCHEMBL7968243

SCHEMBL7968243

O[C@H](COc1cccc2occc12)CN1CCC(O)(c2cnc3ccccc3c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
ABCB1 P08183 10/20 0.47
MAPT P10636 6/20 0.43
TDP1 Q9NUW8 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 2/20 0.42
LMNA P02545 2/20 0.42
ALDH1A1 P00352 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPK1 P28482 3/20 0.42
NPSR1 Q6W5P4 1/20 0.42
DRD2 P14416 3/20 0.41
DRD4 P21917 2/20 0.41
NR1I2 O75469 1/20 0.41
NR3C1 P04150 1/20 0.41
ADRB1 P08588 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968247 0.85 LTA4H (0.38) ABCB1DRD2DRD4HTR1AHTR2A
SCHEMBL7968250 0.84 KCNA3 (0.38) CYP1A2CYP2C19ABCB1DRD2DRD4
SCHEMBL7953370 0.83 HTR1A (0.56) ADRB1HTR1ASLC6A4
SCHEMBL7962648 0.83 ABCB1 (0.47) CYP1A2CYP2C19ABCB1MAPTTDP1
SCHEMBL7953962 0.83 ABCB1 (0.54) CYP1A2CYP2C19ABCB1MAPTTDP1
SCHEMBL7966028 0.82 ABCB1 (0.54) ABCB1MAPTMEN1KMT2ALMNA
SCHEMBL7965524 0.82 ABCB1 (0.48) CYP1A2CYP2C19ABCB1MAPTTDP1
SCHEMBL7953389 0.81 HTR1A (0.53) ABCB1HTR1AADRA2ASLC6A2SLC6A4
SCHEMBL7965363 0.81 PRMT5 (0.48) CYP1A2CYP2C19ABCB1MAPTTDP1
SCHEMBL7969553 0.80 L3MBTL1 (0.55) ABCB1MEN1KMT2AKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed
EP-0976747-A2 Use of 5HT-1F receptor antagonists for treating anxiety disorders ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed