SCHEMBL7953370

SCHEMBL7953370

O[C@H](COc1cccc2[nH]ccc12)CN1CCC(O)(c2cnc3ccccc3c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 19/20 0.56
SLC6A4 P31645 4/20 0.56
ADRB2 P07550 1/20 0.51
ADRB1 P08588 1/20 0.51
ADRB3 P13945 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5584644 0.88 HTR1A (0.59) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7953389 0.86 HTR1A (0.53) HTR1ASLC6A4
SCHEMBL7887623 0.86 ABCB1 (0.61) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7967101 0.86 HTR1A (0.40) HTR1ASLC6A4
SCHEMBL7953373 0.85 HTR1A (0.40) HTR1ASLC6A4ADRB2ADRB1ADRB3
Oxalic Acid SCHEMBL7814401 0.84 HTR1A (0.55) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7953366 0.84 HTR1A (0.43) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7953575 0.83 ADRB2 (0.50) HTR1AADRB2ADRB1ADRB3
SCHEMBL7965169 0.83 ADRB2 (0.50) HTR1AADRB2ADRB1ADRB3
SCHEMBL7814249 0.83 HTR1A (0.58) HTR1ASLC6A4ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed
EP-0976747-A2 Use of 5HT-1F receptor antagonists for treating anxiety disorders ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed