SCHEMBL7968301

SCHEMBL7968301

COc1ccc(Cl)cc1-c1csc(Nc2cccc(-c3ncc[nH]3)c2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.54
PTGS2 P35354 2/20 0.50
MEN1 O00255 5/20 0.48
KMT2A Q03164 5/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 3/20 0.47
CFTR P13569 1/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CYP1A1 P04798 3/20 0.46
CYP1A2 P05177 3/20 0.46
CYP1B1 Q16678 3/20 0.46
GLA P06280 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
PSEN1 P49768 3/20 0.45
PSEN2 P49810 3/20 0.45
APH1B Q8WW43 3/20 0.45
NCSTN Q92542 3/20 0.45
APH1A Q96BI3 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981755 0.84 MAPT (0.64) ALOX5PTGS2MEN1KMT2AMAPT
SCHEMBL7977687 0.83 ALOX5 (0.61) ALOX5PTGS2MEN1KMT2AMAPT
SCHEMBL7968277 0.79 ALOX5 (0.60) ALOX5PTGS2MEN1KMT2APOLB
SCHEMBL3640947 0.79 PSEN1 (0.62) ALOX5PTGS2MEN1KMT2AMAPT
SCHEMBL7967444 0.78 MAPT (0.47) ALOX5PTGS2MEN1KMT2AMAPT
SCHEMBL7129752 0.75 PSEN1 (0.62) ALOX5PTGS2MEN1KMT2APOLB
SCHEMBL12297174 0.75 VCP (0.65) ALOX5PTGS2MEN1KMT2AMAPT
Bromide SCHEMBL7129762 0.74 PSEN1 (0.61) ALOX5PTGS2MEN1KMT2APOLB
SCHEMBL12298012 0.72 KMT2A (0.64) PTGS2MEN1KMT2APOLBMAPT
SCHEMBL3634967 0.72 ALOX5 (0.55) ALOX5PTGS2MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087845-A2 N-CONTAINING HETEROCYCLIC COMPOUNDS AND THEIR USE AS 5-HT ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-22 WO disclosed