SCHEMBL7968588

SCHEMBL7968588

CC(CCC(C#N)(c1ccc(C(F)(F)F)c(C(F)(F)F)c1)C(C)C)N(C)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EBP Q15125 2/20 0.43
SIGMAR1 Q99720 2/20 0.43
KCNH2 Q12809 3/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
HTR2A P28223 2/20 0.39
SLC6A4 P31645 2/20 0.39
ADRA1A P35348 2/20 0.39
SLC6A2 P23975 1/20 0.39
OPRK1 P41145 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CYP3A4 P08684 5/20 0.36
ABCB1 P08183 5/20 0.36
ABCC1 P33527 4/20 0.36
CYP2C19 P33261 2/20 0.36
MEN1 O00255 2/20 0.36
ABCB11 O95342 2/20 0.36
KMT2A Q03164 2/20 0.36
TSHR P16473 2/20 0.36
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7972515 0.90 SIGMAR1 (0.51) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7966287 0.89 EBP (0.41) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7971484 0.89 EBP (0.40) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7968611 0.88 ADRA2B (0.43) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7965746 0.88 SIGMAR1 (0.49) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7965609 0.88 EBP (0.39) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7974383 0.86 SIGMAR1 (0.40) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7956135 0.85 EBP (0.44) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7967090 0.84 ADRA2B (0.41) EBPSIGMAR1KCNH2ADRA2BADRA2C
SCHEMBL7965682 0.84 SIGMAR1 (0.49) EBPSIGMAR1KCNH2ADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed