SCHEMBL7969082

SCHEMBL7969082

CCOC(=O)c1csc(-c2ccc(C(c3cccc(O[Si@H](C)C(C)(C)C)c3)N3C[C@H](C)NC[C@@H]3C)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.38
GAA P10253 1/20 0.38
NPC1 O15118 1/20 0.37
CLK1 P49759 1/20 0.37
OPRD1 P41143 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7969086 0.87 RAB9A (0.38) RAB9AGAANPC1CLK1OPRD1
SCHEMBL7957883 0.86 RAB9A (0.43) RAB9AGAANPC1CLK1OPRD1
SCHEMBL7973745 0.77 OPRD1 (0.45) OPRD1
SCHEMBL7970812 0.74 CYP1A2 (0.48) RAB9AGAAOPRD1CYP1A2CYP3A4
SCHEMBL7967851 0.72 CYP1A2 (0.45) OPRD1CYP1A2CYP3A4
SCHEMBL7968921 0.72 OPRD1 (0.60) OPRD1CYP1A2CYP3A4
SCHEMBL7967499 0.71 RAB9A (0.40) RAB9AGAANPC1CLK1OPRD1
SCHEMBL7957969 0.69 RAB9A (0.48) RAB9AGAANPC1CLK1
SCHEMBL7958101 0.69 RAB9A (0.47) RAB9AGAANPC1CLK1
SCHEMBL7958158 0.68 OPRD1 (0.57) OPRD1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200978-B1 FOR PREVENTING OR TREATING INFLAMMATORY DISEASES SUCH AS ARTHRITIS, PSORIASIS, ASTHMA, OR INFLAMMATORY BOWEL DISEASE, DISORDERS OF RESPIRATORY FUNCTION, GASTROINTESTINAL DISORDERS SUCH AS FUNCTIONAL BOWEL DISEASE, AS ANALGESICS PFIZER INC. 2001-03-13 US disclosed