SCHEMBL7967499

SCHEMBL7967499

CCOC(=O)c1csc(-c2ccc(C(c3cccc(O)c3)N3C[C@@H]4CCCN4C[C@H]3C)cc2)n1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.40
GAA P10253 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CLK1 P49759 2/20 0.39
NPC1 O15118 1/20 0.39
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
PIN1 Q13526 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968609 0.89 PIN1 (0.41) CYP1A2CYP3A4CYP2C9HPGDOPRM1
SCHEMBL7973908 0.88 RAB9A (0.41) RAB9AGAACYP3A4OPRD1CLK1
SCHEMBL7970812 0.85 CYP1A2 (0.48) RAB9AGAACYP1A2CYP3A4CYP2C9
SCHEMBL7957883 0.84 RAB9A (0.43) RAB9AGAACYP1A2CYP3A4CYP2C9
SCHEMBL7967851 0.84 CYP1A2 (0.45) CYP1A2CYP3A4CYP2C9HPGDOPRM1
SCHEMBL7968921 0.83 OPRD1 (0.60) CYP1A2CYP3A4CYP2C9HPGDOPRM1
SCHEMBL7973713 0.76 CYP1A2 (0.48) CYP1A2CYP3A4CYP2C9HPGDOPRM1
SCHEMBL7971327 0.75 CYP1A2 (0.47) CYP1A2CYP3A4CYP2C9HPGDOPRM1
SCHEMBL7971356 0.74
SCHEMBL7968871 0.73 CYP1A2 (0.44) CYP1A2CYP3A4CYP2C9HPGDOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200978-B1 FOR PREVENTING OR TREATING INFLAMMATORY DISEASES SUCH AS ARTHRITIS, PSORIASIS, ASTHMA, OR INFLAMMATORY BOWEL DISEASE, DISORDERS OF RESPIRATORY FUNCTION, GASTROINTESTINAL DISORDERS SUCH AS FUNCTIONAL BOWEL DISEASE, AS ANALGESICS PFIZER INC. 2001-03-13 US disclosed