SCHEMBL7969125

SCHEMBL7969125

Cc1sc(C)c2c1CCCC2(O)c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.32
SIRT2 Q8IXJ6 3/20 0.31
ENPP2 Q13822 1/20 0.30
DRD4 P21917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL769096 0.77 ENPP2 (0.37) ENPP2
SCHEMBL15487989 0.72 CYP11B1 (0.40) SIRT2ENPP2
SCHEMBL26643915 0.70 SIRT2 (0.35) SIRT2ENPP2
SCHEMBL731222 0.69 PGR (0.43) ENPP2DRD4
SCHEMBL31646062 0.68 ENPP2 (0.34) SIRT2ENPP2
SCHEMBL1375313 0.68 HSD11B1 (0.36) SIRT2ENPP2
SCHEMBL7784539 0.67 CYP11B1 (0.40) SIRT2ENPP2DRD4
SCHEMBL7786406 0.67 CYP11B1 (0.40) SIRT2ENPP2DRD4
SCHEMBL29222693 0.67 MAP3K14 (0.38) ENPP2
SCHEMBL7787709 0.67 CYP11B1 (0.37) SIRT2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313309-B1 BENZOTHIOPHENYL-1H-IMIDAZOLE ANALGESICS; HYPOTENSIVE AGENTS, ANTIDEPRESSANTS; SEXUAL, ATTENTION DEFICIT, AND HYPERACTIVE DISORDERS; DELTA-OPIOD RECEPTOR AGONISTS ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-11-06 US disclosed
WO-1999051593-A1 4-THIONAPHTHYL-1H-IMIDAZOLES WITH ALPHA-2-ADRENERGIC ACTIVITY ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 1999-10-14 WO disclosed